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Search results (436 entries covering 174 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
FGFR4FGFRTK6jpjAn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman11051
FGFR4FGFRTK6nvhAAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11388
FGFR4FGFRTK7ybpA~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamideHuman14500
FGFR1FGFRTK7wclAB11-[2,6-bis(fluoranyl)-3,5-dimethoxy-phenyl]-13-ethyl-4-(morpholin-4-ylmethyl)-5,7,11,13-tetrazatricyclo[7.4.0.0^{2,6}]trideca-1(9),2(6),3,7-tetraen-12-oneHuman14363
FGFR4FGFRTK6nviABn-[3-chloro-2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-5-fluorophenyl]propanamideHuman11389
FGFR4FGFRTK4tygAB-Human933
FGFR4FGFRTK4tyiA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman926
FGFR2FGFRTK2pvyCphosphomethylphosphonic acid adenylate esterHuman501
FGFR2FGFRTK8e1xA(5m)-n-methyl-5-{(6m,8s)-5-{[(3s)-oxolan-3-yl]amino}-6-[1-(propan-2-yl)-1h-pyrazol-3-yl]pyrazolo[1,5-a]pyrimidin-3-yl}pyridine-3-carboxamideHuman14511
FGFR4FGFRTK6v9cAAn-[(3r,4s)-4-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}oxolan-3-yl]prop-2-enamideHuman12096
FGFR2FGFRTK7kieBAn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHuman13282
FGFR2FGFRTK6agxCBethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11537
FGFR2FGFRTK6agxABethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11542
FGFR2FGFRTK4j95DAphosphomethylphosphonic acid adenylate esterHuman490
FGFR2FGFRTK4j97DBphosphomethylphosphonic acid adenylate esterHuman532
FGFR2FGFRTK4j96AB-Human470
FGFR2FGFRTK6agxCAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11538
FGFR2FGFRTK4j95BBphosphomethylphosphonic acid adenylate esterHuman519
FGFR2FGFRTK4j95ABphosphomethylphosphonic acid adenylate esterHuman477
FGFR1FGFRTK6itjBB4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHuman11772
FGFR2FGFRTK5ugxABphosphomethylphosphonic acid adenylate esterHuman7448
FGFR2FGFRTK7kiaAB1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHuman13285
FGFR1FGFRTK5flfBA-Human6465
FGFR1FGFRTK5vndAAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHuman7646
FGFR2FGFRTK6v6qCphosphomethylphosphonic acid adenylate esterHuman12969
FGFR2FGFRTK6lvlAn-ethyl-2-[[4-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHuman12132
FGFR2FGFRTK6lvlBn-ethyl-2-[[4-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHuman12130
FGFR1FGFRTK5ew8BB~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHuman6471
FGFR1FGFRTK5a46BB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3578
FGFR1FGFRTK3c4fBB3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHuman3562
FGFR2FGFRTK4j97BAphosphomethylphosphonic acid adenylate esterHuman476
FGFR2FGFRTK6agxBAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11540
FGFR4FGFRTK5nwzA~{n}-[3-[2-(3,5-dimethoxyphenyl)ethyl]-1~{h}-pyrazol-5-yl]-2-(propanoylamino)benzamideHuman9789
FGFR2FGFRTK4j95BAphosphomethylphosphonic acid adenylate esterHuman498
FGFR2FGFRTK4j95CAphosphomethylphosphonic acid adenylate esterHuman531
FGFR2FGFRTK2pwlAphosphomethylphosphonic acid adenylate esterHuman523
FGFR2FGFRTK4j98BBphosphomethylphosphonic acid adenylate esterHuman472
FGFR4FGFRTK4qqcABn-(4-{[3-(3,5-dimethoxyphenyl)-7-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)propanamideHuman932
FGFR2FGFRTK8w38AB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman15403
FGFR2FGFRTK6agxBBethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11536
FGFR2FGFRTK4j97CAphosphomethylphosphonic acid adenylate esterHuman488
FGFR2FGFRTK6lvkBn-ethyl-2-[[4-[[4-(4-methylpiperazin-1-yl)-3-(2-morpholin-4-ylethoxy)phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHuman12129
FGFR2FGFRTK5uglBAphosphoaminophosphonic acid-adenylate esterHuman7450
FGFR1FGFRTK4uwcAB3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHuman6017
FGFR4FGFRTK4qqtA-Human922
FGFR4FGFRTK4qqjA-Human935
FGFR4FGFRTK6jpeAn-[2-[[6-[2-[[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]amino]pyridin-3-yl]pyrimidin-4-yl]amino]-3-methyl-phenyl]prop-2-enamideHuman12230
FGFR4FGFRTK5nudB3-chloranyl-~{n}-(3-nitropyridin-2-yl)-5-(trifluoromethyl)pyridin-2-amineHuman9790
FGFR4FGFRTK7yc3A6-bromanyl-~{n}-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-5-methanoyl-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamideHuman14501
FGFR4FGFRTK4tygAA-Human929
FGFR4FGFRTK6yi8ABn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman12811
FGFR4FGFRTK6yi8BAn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman12813
FGFR4FGFRTK6yi8BBn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman12814
FGFR4FGFRTK6nvjAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-fluorophenyl]propanamideHuman11391
FGFR4FGFRTK5nudA3-chloranyl-~{n}-(3-nitropyridin-2-yl)-5-(trifluoromethyl)pyridin-2-amineHuman9787
FGFR4FGFRTK7vjlAn-[5-(aminomethyl)-4-(2-methoxyethylamino)pyridin-2-yl]-7-[2,2,2-tris(fluoranyl)ethanoyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman14109
FGFR4FGFRTK6nviAAn-[3-chloro-2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-5-fluorophenyl]propanamideHuman11392
FGFR4FGFRTK4r6vAn-[4-({[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino}methyl)phenyl]propanamideHuman931
FGFR4FGFRTK6nvkAAn-[(3s,4s)-3-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}oxan-4-yl]propanamideHuman11395
FGFR4FGFRTK4tyeA-Human927
FGFR4FGFRTK4uxqA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman930
FGFR4FGFRTK5nwzB~{n}-[3-[2-(3,5-dimethoxyphenyl)ethyl]-1~{h}-pyrazol-5-yl]-2-(propanoylamino)benzamideHuman9788
FGFR4FGFRTK4xcuABn-(2-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}-3-methylphenyl)prop-2-enamideHuman924
FGFR4FGFRTK7dtzAn-[2-[[5-[[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]methoxy]pyrimidin-2-yl]amino]-3-methyl-phenyl]-2-fluoranyl-prop-2-enamideHuman13506
FGFR2FGFRTK6v6qBphosphomethylphosphonic acid adenylate esterHuman12966
FGFR2FGFRTK4j99DBphosphomethylphosphonic acid adenylate esterHuman481
FGFR2FGFRTK4j95AAphosphomethylphosphonic acid adenylate esterHuman529
FGFR2FGFRTK4j97BCphosphomethylphosphonic acid adenylate esterHuman510
FGFR2FGFRTK4j97CCphosphomethylphosphonic acid adenylate esterHuman483
FGFR2FGFRTK5ugxBBphosphomethylphosphonic acid adenylate esterHuman7445
FGFR2FGFRTK5uhnBAphosphomethylphosphonic acid adenylate esterHuman7451
FGFR1FGFRTK8jmzAAn-(2-(dimethylamino)ethyl)-1-(3-((4-((2-methyl-1h-indol-5-yl)oxy)pyrimidin-2-yl)amino)phenyl)methanesulfonamideHuman15228
FGFR2FGFRTK6v6qAphosphomethylphosphonic acid adenylate esterHuman12968
FGFR1FGFRTK8jmzABn-(2-(dimethylamino)ethyl)-1-(3-((4-((2-methyl-1h-indol-5-yl)oxy)pyrimidin-2-yl)amino)phenyl)methanesulfonamideHuman15227
FGFR4FGFRTK7v29An-[2-[[3-(3,5-dimethoxyphenyl)-2-oxidanylidene-1-[3-(4-propanoylpiperazin-1-yl)propyl]-4h-pyrimido[4,5-d]pyrimidin-7-yl]amino]phenyl]propanamideHuman14165
FGFR4FGFRTK6iuoAn-({4-[4-amino-3-(3,5-dimethyl-1-benzofuran-2-yl)-7-oxo-6,7-dihydro-2h-pyrazolo[3,4-d]pyridazin-2-yl]phenyl}methyl)prop-2-enamideHuman11757
FGFR2FGFRTK2psqB-Human530
FGFR2FGFRTK2q0bBphosphomethylphosphonic acid adenylate esterHuman499
FGFR2FGFRTK6agxDAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11543
FGFR2FGFRTK2py3Bphosphomethylphosphonic acid adenylate esterHuman484
FGFR2FGFRTK4j95DBphosphomethylphosphonic acid adenylate esterHuman492
FGFR2FGFRTK2pwlBphosphomethylphosphonic acid adenylate esterHuman534
FGFR4FGFRTK4qrcA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman923
FGFR2FGFRTK5uglAAphosphoaminophosphonic acid-adenylate esterHuman7442
FGFR2FGFRTK8u1fAn-[4-(4-amino-7-methyl-5-{4-[(4-methylpyrimidin-2-yl)oxy]phenyl}-7h-pyrrolo[2,3-d]pyrimidin-6-yl)phenyl]-2-methylpropanamideHuman15202
FGFR2FGFRTK5uglBBphosphoaminophosphonic acid-adenylate esterHuman7449
FGFR1FGFRTK5uq0AB2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHuman7458
FGFR3FGFRTK8udvA3-[(6-chloro-1-cyclopropyl-1h-benzimidazol-5-yl)ethynyl]-1-[(3s,5s)-5-(methoxymethyl)-1-(prop-2-enoyl)pyrrolidin-3-yl]-5-(methylamino)-1h-pyrazole-4-carboxamideHuman15203
FGFR3FGFRTK9cd7A(3p)-5-[(1r)-1-(3,5-dichloropyridin-4-yl)ethoxy]-3-{6-[6-(methanesulfonyl)-2,6-diazaspiro[3.3]heptan-2-yl]pyridin-3-yl}-1h-indazoleHuman15469
FGFR3FGFRTK12wwA(2s)-2-{[(6p,8s)-3-chloro-6-(1-{1-[(z)-iminomethyl]piperidin-4-yl}-5-methyl-1h-1,2,3-triazol-4-yl)pyrazolo[1,5-a]pyridin-4-yl]oxy}-2-(5-fluoropyridin-2-yl)ethan-1-olHuman15470
FGFR1FGFRTK43zyAA~{n}-[[(2~{r},3~{s},4~{r},5~{r})-5-[4-azanyl-5-[2-(3,5-dimethoxyphenyl)ethynyl]pyrrolo[2,3-d]pyrimidin-7-yl]-3,4-bis(oxidanyl)oxolan-2-yl]methyl]prop-2-enamideHuman15688
FGFR1FGFRTK43zvA~{n}-[[(2~{r},3~{s},4~{r},5~{r})-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-3,4-bis(oxidanyl)oxolan-2-yl]methyl]prop-2-enamideHuman15689
FGFR1FGFRTK9w1aAxs8148Human15679
FGFR1FGFRTK43zyAB~{n}-[[(2~{r},3~{s},4~{r},5~{r})-5-[4-azanyl-5-[2-(3,5-dimethoxyphenyl)ethynyl]pyrrolo[2,3-d]pyrimidin-7-yl]-3,4-bis(oxidanyl)oxolan-2-yl]methyl]prop-2-enamideHuman15680
FGFR1FGFRTK44ahAAderazantinibHuman15681
FGFR1FGFRTK44adAA2-[5-[2-(3,5-dimethoxyphenyl)ethyl]-1~{h}-pyrazol-3-yl]-6-(4-methylpiperazin-1-yl)-1~{h}-benzimidazoleHuman15682
FGFR1FGFRTK44aaAA(2~{r},3~{s},4~{r},5~{r})-2-[[(azanylidene-$l^{4}-azanylidene)amino]methyl]-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]oxolane-3,4-diolHuman15683
FGFR1FGFRTK43xkAB~{n}-[[(2~{r},3~{s},4~{r},5~{r})-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-3,4-bis(oxidanyl)thiolan-2-yl]methyl]prop-2-enamideHuman15684
FGFR1FGFRTK44acA~{n}-[[(2~{r},3~{s},4~{r},5~{r})-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-3,4-bis(oxidanyl)oxolan-2-yl]methyl]-2-fluoranyl-prop-2-enamideHuman15685
FGFR1FGFRTK9wfkAB(2~{r},3~{r},4~{s},5~{r})-2-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-5-(hydroxymethyl)oxolane-3,4-diolHuman15686
FGFR1FGFRTK9wfkAA(2~{r},3~{r},4~{s},5~{r})-2-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-5-(hydroxymethyl)oxolane-3,4-diolHuman15687
FGFR1FGFRTK9wgtAA(2~{r},3~{s},4~{r},5~{r})-2-(aminomethyl)-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]oxolane-3,4-diolHuman15690
FGFR1FGFRTK9uhiA~{n}-[1-methyl-3-[3-[1-(2-morpholin-4-ylethyl)pyrazol-4-yl]quinoxalin-5-yl]indol-6-yl]propanamideHuman15691
FGFR1FGFRTK9wgtAB(2~{r},3~{s},4~{r},5~{r})-2-(aminomethyl)-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]oxolane-3,4-diolHuman15692
FGFR4FGFRTK7wcwA~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamideHuman14168
FGFR2FGFRTK2pvyAphosphomethylphosphonic acid adenylate esterHuman489
FGFR2FGFRTK4j99BBphosphomethylphosphonic acid adenylate esterHuman495
FGFR2FGFRTK8sweAAn-{4-[4-amino-5-(4-methoxyphenyl)-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl}prop-2-enamideHuman15200
FGFR2FGFRTK5ugxAAphosphomethylphosphonic acid adenylate esterHuman7443
FGFR1FGFRTK2fgiB1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-ureaHuman3541
FGFR1FGFRTK3gqlB(e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanolHuman3506
FGFR1FGFRTK5ur1BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman7969
FGFR1FGFRTK1fgkBB-Human3557
FGFR1FGFRTK5am7AB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3488
FGFR2FGFRTK4j97BBphosphomethylphosphonic acid adenylate esterHuman493
FGFR2FGFRTK5ui0AB-Human7447
FGFR4FGFRTK7yboA~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamideHuman14499
FGFR4FGFRTK5jkgA2-[4-[e-2-[5-[(1r)-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1h-indazol-3-yl]ethenyl]pyrazol-1-yl]ethanolHuman7089
FGFR4FGFRTK6nvkABn-[(3s,4s)-3-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}oxan-4-yl]propanamideHuman11390
FGFR4FGFRTK4qqcAAn-(4-{[3-(3,5-dimethoxyphenyl)-7-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)propanamideHuman934
FGFR4FGFRTK6yi8AAn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman12812
FGFR4FGFRTK9k0jA~{n}-[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]-2-fluoranyl-6-(propanoylamino)benzamideHuman15404
FGFR4FGFRTK6iupABn-{4-[4-amino-3-(3,5-dimethyl-1-benzofuran-2-yl)-7-oxo-6,7-dihydro-2h-pyrazolo[3,4-d]pyridazin-2-yl]phenyl}prop-2-enamideHuman11796
FGFR2FGFRTK6v6qDphosphomethylphosphonic acid adenylate esterHuman12967
FGFR2FGFRTK4j99AAphosphomethylphosphonic acid adenylate esterHuman474
FGFR2FGFRTK8w2xA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]propan-1-oneHuman15406
FGFR2FGFRTK5ui0BBphosphomethylphosphonic acid adenylate esterHuman7440
FGFR2FGFRTK2pz5Aphosphomethylphosphonic acid adenylate esterHuman511
FGFR4FGFRTK6nvgAn-[3,5-dichloro-2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)phenyl]propanamideHuman11394
FGFR2FGFRTK4j99ACphosphomethylphosphonic acid adenylate esterHuman469
FGFR2FGFRTK4j99CBphosphomethylphosphonic acid adenylate esterHuman506
FGFR2FGFRTK5eg3Aphosphomethylphosphonic acid adenylate esterHuman6368
FGFR2FGFRTK2pvfAphosphomethylphosphonic acid adenylate esterHuman525
FGFR2FGFRTK5uhnABphosphomethylphosphonic acid adenylate esterHuman7441
FGFR2FGFRTK9u3nA~{n}-[4-[4-azanyl-7-methyl-5-[2-(3-methylimidazo[4,5-b]pyridin-6-yl)ethynyl]pyrrolo[2,3-d]pyrimidin-6-yl]phenyl]prop-2-enamideHuman15407
FGFR2FGFRTK4j97AAphosphomethylphosphonic acid adenylate esterHuman496
FGFR2FGFRTK2pz5Bphosphomethylphosphonic acid adenylate esterHuman513
FGFR2FGFRTK2pzpBphosphomethylphosphonic acid adenylate esterHuman524
FGFR2FGFRTK4j98AB-Human475
FGFR2FGFRTK4j98BAphosphomethylphosphonic acid adenylate esterHuman516
FGFR2FGFRTK2pvyDphosphomethylphosphonic acid adenylate esterHuman482
FGFR2FGFRTK7ozyAA4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman13999
FGFR2FGFRTK5uhnBBphosphomethylphosphonic acid adenylate esterHuman7444
FGFR2FGFRTK4j99BAphosphomethylphosphonic acid adenylate esterHuman518
FGFR2FGFRTK5uglABphosphoaminophosphonic acid-adenylate esterHuman7452
FGFR2FGFRTK6lvkAn-ethyl-2-[[4-[[4-(4-methylpiperazin-1-yl)-3-(2-morpholin-4-ylethoxy)phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHuman12131
FGFR2FGFRTK4j96BBphosphomethylphosphonic acid adenylate esterHuman486
FGFR2FGFRTK8w3bAA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman15408
FGFR2FGFRTK6agxDBethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11539
FGFR2FGFRTK2pzrAphosphomethylphosphonic acid adenylate esterHuman526
FGFR2FGFRTK8w3dAB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman15409
FGFR2FGFRTK4j99DAphosphomethylphosphonic acid adenylate esterHuman533
FGFR2FGFRTK1gjoA-Human478
FGFR2FGFRTK4j99CCphosphomethylphosphonic acid adenylate esterHuman471
FGFR2FGFRTK7kiaAA1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHuman13283
FGFR2FGFRTK5ugxBAphosphomethylphosphonic acid adenylate esterHuman7454
FGFR2FGFRTK2pzpAphosphomethylphosphonic acid adenylate esterHuman497
FGFR2FGFRTK7kieBBn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHuman13284
FGFR2FGFRTK4j96AA-Human473
FGFR2FGFRTK9vlmA~{n}-[3-[2-[[3-[2-(dimethylamino)ethylsulfamoylmethyl]phenyl]amino]pyrimidin-4-yl]-1-methyl-indol-6-yl]propanamideHuman15413
FGFR2FGFRTK7kieABn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHuman13286
FGFR2FGFRTK2pvyBphosphomethylphosphonic acid adenylate esterHuman504
FGFR2FGFRTK7kieAAn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHuman13287
FGFR2FGFRTK7kiaBB1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHuman13288
FGFR2FGFRTK6agxAAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11541
FGFR1FGFRTK5flfDA-Human6468
FGFR3FGFRTK6pnxAAphosphomethylphosphonic acid adenylate esterHuman11948
FGFR3FGFRTK6lvmA2-[[5-[2-(3,5-dimethoxyphenyl)ethyl]-2-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]pyrimidin-4-yl]amino]-n-ethyl-benzenesulfonamideHuman12134
FGFR3FGFRTK6pnxABphosphomethylphosphonic acid adenylate esterHuman11946
FGFR4FGFRTK7wcxA~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamideHuman14166
FGFR2FGFRTK4j96BAphosphomethylphosphonic acid adenylate esterHuman485
FGFR4FGFRTK7f3mA6-[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]-2-(methylamino)-8-[3-(4-prop-2-enoylpiperazin-1-yl)propyl]pyrido[2,3-d]pyrimidin-7-oneHuman14034
FGFR2FGFRTK8h75A4-[9-(2-chlorophenyl)-6-methyl-2,4,5,8,12-pentazatricyclo[8.4.0.0^{3,7}]tetradeca-1(10),3,6,8,11,13-hexaen-13-yl]morpholineHuman14860
FGFR3FGFRTK7dhlA5-[2-(3,5-dimethoxyphenyl)ethyl]-n-[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]pyrimidin-2-amineHuman13258
FGFR3FGFRTK4k33ABphosphomethylphosphonic acid adenylate esterHuman1870
FGFR3FGFRTK6pnxBBphosphomethylphosphonic acid adenylate esterHuman11949
FGFR3FGFRTK4k33AAphosphomethylphosphonic acid adenylate esterHuman1871
FGFR3FGFRTK6pnxBAphosphomethylphosphonic acid adenylate esterHuman11947
FGFR3FGFRTK8uduAB3-[(6-chloro-1-cyclopropyl-1h-benzimidazol-5-yl)ethynyl]-1-[(3s,5s)-5-(methoxymethyl)-1-(prop-2-enoyl)pyrrolidin-3-yl]-5-(methylamino)-1h-pyrazole-4-carboxamideHuman15204
FGFR2FGFRTK3ri1B(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHuman528
FGFR4FGFRTK6iupAAn-{4-[4-amino-3-(3,5-dimethyl-1-benzofuran-2-yl)-7-oxo-6,7-dihydro-2h-pyrazolo[3,4-d]pyridazin-2-yl]phenyl}prop-2-enamideHuman11797
FGFR4FGFRTK4qq5An-(4-{[3-(3,5-dimethoxyphenyl)-7-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)propanamideHuman921
FGFR1FGFRTK5uq0AA2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHuman7456
FGFR1FGFRTK4rwlB6-({7-[(1-aminocyclopropyl)methoxy]-6-methoxyquinolin-4-yl}oxy)-n-methylnaphthalene-1-carboxamideHuman3596
FGFR1FGFRTK6mzwBA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11165
FGFR1FGFRTK3rhxB(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHuman3522
FGFR1FGFRTK4zsaAA4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman3491
FGFR1FGFRTK6c1bBB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11167
FGFR1FGFRTK4rwjBBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3559
FGFR1FGFRTK4v05ABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3593
FGFR1FGFRTK5z0sBB1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHuman10814
FGFR1FGFRTK44adAB2-[5-[2-(3,5-dimethoxyphenyl)ethyl]-1~{h}-pyrazol-3-yl]-6-(4-methylpiperazin-1-yl)-1~{h}-benzimidazoleHuman15672
FGFR1FGFRTK3tt0BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHuman3547
FGFR1FGFRTK1agwBB3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHuman3510
FGFR1FGFRTK8jqiB-Human15678
FGFR1FGFRTK5vndBAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHuman7647
FGFR1FGFRTK7ozdAAn-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]benzamideHuman14007
FGFR1FGFRTK5am7AA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3533
FGFR1FGFRTK6mzqBB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11171
FGFR1FGFRTK6nvlDBn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11398
FGFR1FGFRTK6p69BAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHuman11331
FGFR1FGFRTK5zv2B4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamideHuman10054
FGFR1FGFRTK4v04AA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3542
FGFR1FGFRTK4uwyAB-Human3582
FGFR1FGFRTK5a46BA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3526
FGFR1FGFRTK5uq0BA2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHuman7459
FGFR1FGFRTK4f65BA5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHuman3545
FGFR1FGFRTK1fgkBA-Human3513
FGFR1FGFRTK6c18AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11168
FGFR1FGFRTK1agwAA3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHuman3520
FGFR1FGFRTK5a4cAA1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHuman3543
FGFR1FGFRTK4nk9Bn~4~-{5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3535
FGFR1FGFRTK7ozbAB4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman14008
FGFR1FGFRTK5ur1BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman7971
FGFR1FGFRTK4uwyBA-Human3537
FGFR1FGFRTK4f64BA5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3576
FGFR1FGFRTK4rwkABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3517
FGFR1FGFRTK1fgiAA3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHuman3555
FGFR1FGFRTK3c4fAA3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHuman3515
FGFR1FGFRTK6c19AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11163
FGFR1FGFRTK3ky2A-Human3534
FGFR1FGFRTK5am6BB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3521
FGFR1FGFRTK5o4aAA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHuman9554
FGFR1FGFRTK4rwiBB-Human3527
FGFR1FGFRTK5flfCB-Human6466
FGFR1FGFRTK5a4cBB1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHuman3540
FGFR1FGFRTK5o4aAB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHuman9558
FGFR1FGFRTK6c1oAAn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHuman11159
FGFR1FGFRTK5b7vA[5-amino-1-(2-methyl-1h-benzimidazol-6-yl)-1h-pyrazol-4-yl](1h-indol-2-yl)methanoneHuman6705
FGFR1FGFRTK4nkaAn~4~-{3-[2-(3,4-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3501
FGFR1FGFRTK4zsaBB4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman3512
FGFR1FGFRTK6mzwAB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11157
FGFR1FGFRTK6mzqAB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11156
FGFR1FGFRTK6itjBA4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHuman11775
FGFR1FGFRTK4f64AB5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3589
FGFR1FGFRTK4uwcAA3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHuman6019
FGFR1FGFRTK3tt0BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHuman3581
FGFR1FGFRTK4rwlA-Human3516
FGFR1FGFRTK3c4fAB3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHuman3564
FGFR1FGFRTK5am6AA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3494
FGFR1FGFRTK6mzwBB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman10857
FGFR1FGFRTK5am7BB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3531
FGFR1FGFRTK6itjAA4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHuman11773
FGFR1FGFRTK6c19AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10859
FGFR1FGFRTK5flfCA-Human6469
FGFR1FGFRTK6nvlBAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11403
FGFR1FGFRTK7ozbAA4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman14010
FGFR1FGFRTK5ur1AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman7970
FGFR1FGFRTK6c1bAA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11169
FGFR1FGFRTK3gqiAphosphomethylphosphonic acid adenylate esterHuman3566
FGFR1FGFRTK4v05BAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3518
FGFR1FGFRTK7ozfAAn-[6-(3-ethoxyphenyl)-1h-indazol-3-yl]benzamideHuman14011
FGFR1FGFRTK4rwiAB-Human3551
FGFR1FGFRTK6nvlABn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11401
FGFR1FGFRTK3gqlA(e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanolHuman3509
FGFR1FGFRTK6c19BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10855
FGFR1FGFRTK6c1bAB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10861
FGFR1FGFRTK6p69ABn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHuman11330
FGFR4FGFRTK8kh9A1-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-3-[6-methanoyl-5-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3-(2-morpholin-4-ylethoxy)pyridin-2-yl]ureaHuman15284
FGFR4FGFRTK8kh7A1-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-3-[6-methanoyl-5-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3-(2-morpholin-4-ylethoxy)pyridin-2-yl]ureaHuman15286
FGFR4FGFRTK8kh6A1-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-3-[5-bromanyl-6-(hydroxymethyl)-3-methoxy-pyridin-2-yl]ureaHuman15287
FGFR4FGFRTK8w5cAn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-5-methanoyl-6-[(4-methylpiperazin-1-yl)methyl]-1-propan-2-yl-pyrrolo[3,2-b]pyridine-3-carboxamideHuman15288
FGFR4FGFRTK4tyjA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman925
FGFR4FGFRTK6nvhABn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11393
FGFR2FGFRTK3ri1A(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHuman503
FGFR2FGFRTK8stgAn-{4-[(5p)-4-amino-5-{3-fluoro-4-[(4-methylpyrimidin-2-yl)oxy]phenyl}-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl}-2-methylprop-2-enamideHuman14762
FGFR2FGFRTK4j98AA-Human500
FGFR4FGFRTK5xfjA2-[4-[e-2-[5-[(1r)-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1h-indazol-3-yl]ethenyl]pyrazol-1-yl]ethanolHuman10376
FGFR1FGFRTK4v01AB3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3590
FGFR2FGFRTK4j97ABphosphomethylphosphonic acid adenylate esterHuman527
FGFR2FGFRTK8sweABn-{4-[4-amino-5-(4-methoxyphenyl)-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl}prop-2-enamideHuman15201
FGFR2FGFRTK4j99ABphosphomethylphosphonic acid adenylate esterHuman494
FGFR2FGFRTK5ui0BAphosphomethylphosphonic acid adenylate esterHuman7453
FGFR1FGFRTK4rwkAAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3500
FGFR1FGFRTK5am6BA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3587
FGFR1FGFRTK6mzqAA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman10860
FGFR1FGFRTK3js2B5-(2-thienyl)nicotinic acidHuman3504
FGFR1FGFRTK6c1oBBn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHuman11154
FGFR1FGFRTK4f63A5-bromo-n~4~-(3-methyl-1h-pyrazol-5-yl)-n~2~-[2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamineHuman3563
FGFR1FGFRTK3js2A5-(2-thienyl)nicotinic acidHuman3523
FGFR1FGFRTK1agwAB3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHuman3528
FGFR1FGFRTK6mzwAA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11162
FGFR1FGFRTK1fgkAB-Human3546
FGFR1FGFRTK4v04AB-Human3571
FGFR1FGFRTK4uwyAA-Human3489
FGFR1FGFRTK6nvlCBn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11405
FGFR1FGFRTK3ky2B-Human3525
FGFR1FGFRTK6p68Bn-{3-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-1-(2-hydroxyethyl)-1h-pyrazol-4-yl}prop-2-enamideHuman11334
FGFR1FGFRTK4rwjABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3519
FGFR1FGFRTK5flfEB-Human6472
FGFR1FGFRTK6c1bBA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10856
FGFR1FGFRTK4uwcBA3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHuman6021
FGFR1FGFRTK4nksABn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHuman3561
FGFR1FGFRTK4v01BB3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3594
FGFR1FGFRTK4f65BB5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHuman3502
FGFR1FGFRTK7wclAA11-[2,6-bis(fluoranyl)-3,5-dimethoxy-phenyl]-13-ethyl-4-(morpholin-4-ylmethyl)-5,7,11,13-tetrazatricyclo[7.4.0.0^{2,6}]trideca-1(9),2(6),3,7-tetraen-12-oneHuman14364
FGFR1FGFRTK5a46AB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3505
FGFR1FGFRTK6c1cAB7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10853
FGFR1FGFRTK4wunAAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3511
FGFR4FGFRTK8kh8A1-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-3-[6-methanoyl-5-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3-(2-morpholin-4-ylethoxy)pyridin-2-yl]ureaHuman15285
FGFR1FGFRTK6itjAB4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHuman11774
FGFR1FGFRTK6nvlDAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11402
FGFR1FGFRTK3rhxA(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHuman3554
FGFR1FGFRTK5ew8AB~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHuman6461
FGFR1FGFRTK4rwiBA-Human3569
FGFR1FGFRTK5flfDB-Human6463
FGFR1FGFRTK4f65AB5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHuman3508
FGFR1FGFRTK4wunBBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3565
FGFR4FGFRTK7yc1A~{n}-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-5-methanoyl-1-propyl-pyrrolo[3,2-b]pyridine-3-carboxamideHuman14498
FGFR4FGFRTK7ybxA~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamideHuman14502
FGFR4FGFRTK6v9cABn-[(3r,4s)-4-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}oxolan-3-yl]prop-2-enamideHuman12095
FGFR4FGFRTK9k0iA(2~{s})-~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]-2-cyano-3-cyclopropyl-propanamideHuman15405
FGFR4FGFRTK4xcuAAn-(2-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}-3-methylphenyl)prop-2-enamideHuman928
FGFR4FGFRTK7wctA~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamideHuman14167
FGFR4FGFRTK5xffA2-[4-[e-2-[5-[(1r)-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1h-indazol-3-yl]ethenyl]pyrazol-1-yl]ethanolHuman10375
FGFR2FGFRTK7kiaBA1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHuman13281
FGFR2FGFRTK1oecA4-aryl-2-phenylamino pyrimidineHuman479
FGFR2FGFRTK4j95CBphosphomethylphosphonic acid adenylate esterHuman502
FGFR2FGFRTK2py3Aphosphomethylphosphonic acid adenylate esterHuman509
FGFR2FGFRTK3clyAphosphomethylphosphonic acid adenylate esterHuman522
FGFR2FGFRTK7ozyAB4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman13998
FGFR2FGFRTK4j99CAphosphomethylphosphonic acid adenylate esterHuman505
FGFR2FGFRTK4j99DCphosphomethylphosphonic acid adenylate esterHuman480
FGFR2FGFRTK4j99BCphosphomethylphosphonic acid adenylate esterHuman491
FGFR2FGFRTK2psqA-Human515
FGFR2FGFRTK2pzrBphosphomethylphosphonic acid adenylate esterHuman508
FGFR2FGFRTK5ui0AA-Human7446
FGFR2FGFRTK2q0bAphosphomethylphosphonic acid adenylate esterHuman512
FGFR2FGFRTK5uhnAAphosphomethylphosphonic acid adenylate esterHuman7455
FGFR2FGFRTK4j97DAphosphomethylphosphonic acid adenylate esterHuman507
FGFR2FGFRTK8w3dAA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman15410
FGFR2FGFRTK4j97ACphosphomethylphosphonic acid adenylate esterHuman521
FGFR2FGFRTK3b2tA5'-o-[(s)-hydroxy{[(s)-hydroxy(methyl)phosphoryl]oxy}phosphoryl]adenosineHuman520
FGFR2FGFRTK8w38AA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman15411
FGFR2FGFRTK3b2tB5'-o-[(s)-hydroxy{[(s)-hydroxy(methyl)phosphoryl]oxy}phosphoryl]adenosineHuman517
FGFR2FGFRTK8w3bAB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman15412
FGFR2FGFRTK4j97CBphosphomethylphosphonic acid adenylate esterHuman487
FGFR2FGFRTK4j97DCphosphomethylphosphonic acid adenylate esterHuman514
FGFR2FGFRTK10ooA(4p)-n-[4-(4-aminopiperidin-1-yl)-2-methoxyphenyl]-5-chloro-4-(1h-indol-3-yl)pyrimidin-2-amineHuman15414
FGFR3FGFRTK8uduAA3-[(6-chloro-1-cyclopropyl-1h-benzimidazol-5-yl)ethynyl]-1-[(3s,5s)-5-(methoxymethyl)-1-(prop-2-enoyl)pyrrolidin-3-yl]-5-(methylamino)-1h-pyrazole-4-carboxamideHuman15205
FGFR3FGFRTK8udtA3-[(1-cyclopropyl-4,6-difluoro-1h-benzimidazol-5-yl)ethynyl]-1-[(3r,5r)-5-(methoxymethyl)-1-propanoylpyrrolidin-3-yl]-5-(methylamino)-1h-pyrazole-4-carboxamideHuman15206
FGFR1FGFRTK6nvlCAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11404
FGFR1FGFRTK4wunABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3595
FGFR1FGFRTK4nksBAn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHuman3492
FGFR1FGFRTK3kxxD-Human3503
FGFR1FGFRTK44aaAB(2~{r},3~{s},4~{r},5~{r})-2-[[(azanylidene-$l^{4}-azanylidene)amino]methyl]-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]oxolane-3,4-diolHuman15671
FGFR1FGFRTK5o4aBB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHuman9555
FGFR1FGFRTK5z0sBA1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHuman10812
FGFR1FGFRTK6nvlAAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11400
FGFR1FGFRTK5b7vB[5-amino-1-(2-methyl-1h-benzimidazol-6-yl)-1h-pyrazol-4-yl](1h-indol-2-yl)methanoneHuman6704
FGFR1FGFRTK7ozfABn-[6-(3-ethoxyphenyl)-1h-indazol-3-yl]benzamideHuman14006
FGFR1FGFRTK4v05BBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3493
FGFR1FGFRTK4v01AA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3556
FGFR1FGFRTK5am7BA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3588
FGFR1FGFRTK5flfBB-Human6467
FGFR1FGFRTK6p68An-{3-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-1-(2-hydroxyethyl)-1h-pyrazol-4-yl}prop-2-enamideHuman11336
FGFR1FGFRTK5flfEA-Human6473
FGFR1FGFRTK5o49BB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHuman9557
FGFR1FGFRTK6p68Cn-{3-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-1-(2-hydroxyethyl)-1h-pyrazol-4-yl}prop-2-enamideHuman11332
FGFR1FGFRTK4rwkBAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3591
FGFR1FGFRTK5ew8BA~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHuman6474
FGFR1FGFRTK5am6AB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3514
FGFR1FGFRTK5o49AA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHuman9560
FGFR1FGFRTK4f65AA5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHuman3558
FGFR1FGFRTK4nk9An~4~-{5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3550
FGFR1FGFRTK5flfAA-Human6462
FGFR1FGFRTK9vljA~{n}-[3-[2-[[3-[2-(dimethylamino)ethylsulfamoylmethyl]phenyl]amino]pyrimidin-4-yl]-1-methyl-indol-6-yl]propanamideHuman15673
FGFR1FGFRTK3kxxB-Human3575
FGFR1FGFRTK5o4aBA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHuman9559
FGFR1FGFRTK4uwbABn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHuman6023
FGFR1FGFRTK43xkAA~{n}-[[(2~{r},3~{s},4~{r},5~{r})-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-3,4-bis(oxidanyl)thiolan-2-yl]methyl]prop-2-enamideHuman15674
FGFR1FGFRTK1fgkAA-Human3592
FGFR1FGFRTK6nvlBBn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11399
FGFR1FGFRTK6mzqBA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11161
FGFR1FGFRTK6c19BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10862
FGFR1FGFRTK9u7gA(e)-4-methyl-17-(1-methyl-1h-pyrazol-4-yl)-7,10-dioxa-4-aza-1(3,6)-imidazo[1,2-b]pyridazina-2(3,5)-pyridinacyclodecaphan-3-oneHuman15675
FGFR1FGFRTK5a4cAB1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHuman3498
FGFR1FGFRTK6c1oBAn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHuman11160
FGFR1FGFRTK1fgiBA3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHuman3586
FGFR1FGFRTK6c1cBB7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11158
FGFR1FGFRTK6c18BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10854
FGFR1FGFRTK9uhcA~{n}-[1-methyl-3-[2-[1-(2-morpholin-4-ylethyl)pyrazol-4-yl]-5~{h}-pyrrolo[2,3-b]pyrazin-7-yl]indol-6-yl]propanamideHuman15676
FGFR1FGFRTK44ahABderazantinibHuman15677
FGFR1FGFRTK6c1cAA7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11164
FGFR1FGFRTK5ew8AA~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHuman6470
FGFR1FGFRTK4f64BB5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3553
FGFR1FGFRTK5zv2A4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamideHuman10055
FGFR1FGFRTK5o49AB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHuman9556
FGFR1FGFRTK4f63B5-bromo-n~4~-(3-methyl-1h-pyrazol-5-yl)-n~2~-[2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamineHuman3574
FGFR1FGFRTK3tt0AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHuman3567
FGFR1FGFRTK5o49BA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHuman9561
FGFR1FGFRTK4wunBAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3529
FGFR1FGFRTK1fgiAB3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHuman3552
FGFR1FGFRTK4f64AA5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3548
FGFR1FGFRTK5vndBBn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHuman7645
FGFR1FGFRTK4uwbBAn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHuman6018
FGFR1FGFRTK3c4fBA3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHuman3573
FGFR1FGFRTK4rwjAAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3584
FGFR1FGFRTK4rwkBBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3530
FGFR1FGFRTK4zsaAB4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman3487
FGFR1FGFRTK4v01BA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3497
FGFR1FGFRTK4uwbBBn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHuman6022
FGFR1FGFRTK3tt0AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHuman3538
FGFR1FGFRTK4nksAAn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHuman3570
FGFR1FGFRTK4nksBBn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHuman3577
FGFR1FGFRTK4rwjBAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3579
FGFR1FGFRTK4zsaBA4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman3572
FGFR1FGFRTK3kxxA-Human3495
FGFR1FGFRTK4v04BB-Human3496
FGFR1FGFRTK1agwBA3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHuman3568
FGFR1FGFRTK5a4cBA1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHuman3585
FGFR1FGFRTK5vndABn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHuman7648
FGFR1FGFRTK5z0sAA1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHuman10813
FGFR1FGFRTK6c18BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11170
FGFR1FGFRTK5flfAB-Human6464
FGFR1FGFRTK5z0sAB1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHuman10815
FGFR1FGFRTK4nkaBn~4~-{3-[2-(3,4-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3539
FGFR1FGFRTK4uwbAAn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHuman6020
FGFR1FGFRTK5a46AA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3532
FGFR1FGFRTK6c1oABn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHuman11166
FGFR1FGFRTK3kxxC-Human3549
FGFR1FGFRTK2fgiA1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-ureaHuman3490
FGFR1FGFRTK7ozdABn-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]benzamideHuman14009
FGFR1FGFRTK3gqlC(e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanolHuman3536
FGFR1FGFRTK5ur1AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman7972
FGFR1FGFRTK1fgiBB3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHuman3580
FGFR1FGFRTK4rwiAA-Human3499
FGFR1FGFRTK6c1cBA7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10858
FGFR1FGFRTK6p69AAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHuman11333
FGFR1FGFRTK6p69BBn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHuman11335
FGFR1FGFRTK4v04BA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3524
FGFR1FGFRTK4v05AAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3560
FGFR1FGFRTK4uwyBB-Human3583
FGFR1FGFRTK5uq0BB2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHuman7457
FGFR1FGFRTK4uwcBB3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHuman6016
FGFR1FGFRTK6c18AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11155
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