Searching for structures with analogs of Belumosudil.

Search results (10 entries covering 5 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetailsSimilarity (MFP)File
MELKCAMKLCAMK9f31An-[4-(1h-indazol-5-yl)phenyl]propanamideHuman157870.43
ULK1ULKOther9f32AAn-[4-(1h-indazol-5-yl)phenyl]propanamideHuman155450.43
TGFBR1 (TGFbR1)STKRTKL3gxlAn-1h-indazol-5-yl-2-(6-methylpyridin-2-yl)quinazolin-4-amineHuman21160.56
ULK1ULKOther9f32ABn-[4-(1h-indazol-5-yl)phenyl]propanamideHuman155480.43
CAMK1D (CaMK1d)CAMK1CAMK2jc6CAn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman48320.42
CAMK1D (CaMK1d)CAMK1CAMK2jc6CBn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman48310.42
CAMK1D (CaMK1d)CAMK1CAMK2jc6ABn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman48300.42
CAMK1D (CaMK1d)CAMK1CAMK2jc6AAn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman48290.42
CSNK2A1 (CK2a1)CK2CMGC7z39AB2-[3-[4-(1~{h}-indazol-5-ylamino)quinazolin-2-yl]phenoxy]-~{n}-propan-2-yl-ethanamideHuman144451.00
CSNK2A1 (CK2a1)CK2CMGC7z39AA2-[3-[4-(1~{h}-indazol-5-ylamino)quinazolin-2-yl]phenoxy]-~{n}-propan-2-yl-ethanamideHuman144491.00