Searching for structures with analogs of Belumosudil.
Search results (10 entries covering 5 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | Similarity (MFP) | File |
|---|---|---|---|---|---|---|---|---|---|---|---|
| MELK | CAMKL | CAMK | 9f31 | A | n-[4-(1h-indazol-5-yl)phenyl]propanamide | Human | 15787 | 0.43 | |||
| ULK1 | ULK | Other | 9f32 | A | A | n-[4-(1h-indazol-5-yl)phenyl]propanamide | Human | 15545 | 0.43 | ||
| TGFBR1 (TGFbR1) | STKR | TKL | 3gxl | A | n-1h-indazol-5-yl-2-(6-methylpyridin-2-yl)quinazolin-4-amine | Human | 2116 | 0.56 | |||
| ULK1 | ULK | Other | 9f32 | A | B | n-[4-(1h-indazol-5-yl)phenyl]propanamide | Human | 15548 | 0.43 | ||
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 2jc6 | C | A | n-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amine | Human | 4832 | 0.42 | ||
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 2jc6 | C | B | n-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amine | Human | 4831 | 0.42 | ||
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 2jc6 | A | B | n-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amine | Human | 4830 | 0.42 | ||
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 2jc6 | A | A | n-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amine | Human | 4829 | 0.42 | ||
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7z39 | A | B | 2-[3-[4-(1~{h}-indazol-5-ylamino)quinazolin-2-yl]phenoxy]-~{n}-propan-2-yl-ethanamide | Human | 14445 | 1.00 | ||
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7z39 | A | A | 2-[3-[4-(1~{h}-indazol-5-ylamino)quinazolin-2-yl]phenoxy]-~{n}-propan-2-yl-ethanamide | Human | 14449 | 1.00 |