Searching for structures with analogs of -.
Search results (10 entries covering 6 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | Similarity (MFP) | File |
|---|---|---|---|---|---|---|---|---|---|---|---|
| PIM1 | PIM | CAMK | 2c3i | B | A | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 2348 | 0.51 | ||
| PIM1 | PIM | CAMK | 2c3i | B | B | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 2374 | 0.51 | ||
| PIM1 | PIM | CAMK | 3bgq | A | n-cyclohexyl-3-[3-(trifluoromethyl)phenyl][1,2,4]triazolo[4,3-b]pyridazin-6-amine | Human | 2465 | 0.62 | |||
| CLK1 | CLK | CMGC | 6yta | A | B | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 12417 | 0.51 | ||
| CLK1 | CLK | CMGC | 6yta | A | A | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 12423 | 0.51 | ||
| ACVR1 (ALK2) | STKR | TKL | 4dym | A | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 1509 | 0.51 | |||
| ACVR1 (ALK2) | STKR | TKL | 3oom | A | A | 1-{3-[6-(tetrahydro-2h-pyran-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}ethanone | Human | 1517 | 0.55 | ||
| ACVR1 (ALK2) | STKR | TKL | 3oom | A | B | 1-{3-[6-(tetrahydro-2h-pyran-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}ethanone | Human | 1518 | 0.55 | ||
| HASPIN (Haspin) | Haspin | Other | 3f2n | A | B | (2s)-2-{[3-(3-aminophenyl)imidazo[1,2-b]pyridazin-6-yl]amino}-3-methylbutan-1-ol | Human | 3813 | 0.40 | ||
| HASPIN (Haspin) | Haspin | Other | 3f2n | A | A | (2s)-2-{[3-(3-aminophenyl)imidazo[1,2-b]pyridazin-6-yl]amino}-3-methylbutan-1-ol | Human | 3803 | 0.40 |