Searching for structures with analogs of Trametinib.
Search results (2 entries covering 1 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | Similarity (MFP) | File |
|---|---|---|---|---|---|---|---|---|---|---|---|
| MAP2K1 | STE7 | STE | 9ecu | B | A | 4-[2-chloro-3-(methylsulfamamido)phenoxy]-n-cyclopropyl-2-(2-fluoro-4-iodoanilino)-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide | Human | 16172 | 0.42 | ||
| MAP2K1 | STE7 | STE | 9ecu | B | B | 4-[2-chloro-3-(methylsulfamamido)phenoxy]-n-cyclopropyl-2-(2-fluoro-4-iodoanilino)-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide | Human | 16174 | 0.42 |